N-[5-(1-邻氯苯氧乙基)-1,3,4-噻二唑-2-基]-N'- 芳氧乙酰基硫脲的合成与生物活性

王子云; 王胜; 宋新建; 汪焱钢

N-[5-(1-邻氯苯氧乙基)-1,3,4-噻二唑-2-基]-N'- 芳氧乙酰基硫脲的合成与生物活性

1.
周口师范学院化学系,河南周口 466000
2.
华中师范大学化学学院,湖北武汉 430079

基金项目:

国家自然科学基金(20072009)资助项目.

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出版历程
- 收稿日期: 2005-03-23

Synthesis and Biological Activity of N[5-(1-o-Chlorophenoxyethyl)-1,3,4-thiodiazol-2-yl]- N'- aryloxyacetyl Thioureas

1.
Department of Chemistry,Zhoukou Normal University, Zhoukou 466000,China
2.
College of Chemistry,Central China Normal University, Wuhan 430079,China

摘要

摘要: 为了寻找新的高生物活性农药,通过2-氨基-5-(1-邻氯苯氧乙基)-1,3,4-噻二唑与芳氧乙酰基异硫氰酸酯反应,合成了9个新的芳氧乙酰基硫脲,初步的生物活性测定结果表明,部分目标化合物具有良好的植物生长调节活性,其中 2c、2d 具有较好的生长素活性,其生长促进率分别为26.9%和27.2%。
- 酰基硫脲 /
- 1,3,4 -噻二唑 /
- 合成 /
- 生物活性 /
- 生长素
Abstract: In order to search for high biological active pesticide, nine novel aryloxyacetyl thioureas have been synthesized by the reaction of 2-amino-5-(1-o-chlorophenoxyethyl)-1,3,4-thiodiazole with aryloxyacetyl isothiocyanates. The preliminary biological activity tests exhibited that some target compounds possessed a good activity as plant growth regulator, and 2c and 2d had better activities as auxin, the promoting rate were 26.9% and 27.2%.
- acyl thiourea /
- 1,3,4-thiodiazole /
- synthesis /
- bioactivity /
- auxin

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参考文献(9)

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