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2-溴代呋喃基或噻吩基-1,3-二噻烷衍生物的合成及杀虫活性

王磊 孙薇 鲁东飞 柳明 段又生王敏 刘尚钟

王磊, 孙薇, 鲁东飞, 柳明, 段又生王敏, 刘尚钟. 2-溴代呋喃基或噻吩基-1,3-二噻烷衍生物的合成及杀虫活性[J]. 农药学学报, 2008, 10(2): 147-150.
引用本文: 王磊, 孙薇, 鲁东飞, 柳明, 段又生王敏, 刘尚钟. 2-溴代呋喃基或噻吩基-1,3-二噻烷衍生物的合成及杀虫活性[J]. 农药学学报, 2008, 10(2): 147-150.
WANG Lei, SUN Wei, LU Dong-fei, LIU Ming, DUAN You-sheng, WANG Min. Synthesis and Insecticidal Activity of 2--1,3-dithiane Derivatives(Department of Applied Chemistry,China Agricultural University,Key Laboratory of PesticideChemistry and Application Technology,Beijing 100193,China)[J]. Chinese Journal of Pesticide Science, 2008, 10(2): 147-150.
Citation: WANG Lei, SUN Wei, LU Dong-fei, LIU Ming, DUAN You-sheng, WANG Min. Synthesis and Insecticidal Activity of 2--1,3-dithiane Derivatives(Department of Applied Chemistry,China Agricultural University,Key Laboratory of PesticideChemistry and Application Technology,Beijing 100193,China)[J]. Chinese Journal of Pesticide Science, 2008, 10(2): 147-150.

2-溴代呋喃基或噻吩基-1,3-二噻烷衍生物的合成及杀虫活性

基金项目: 

国家自然科学基金资助项目(20572129);国家"十一五"科技支撑计划项目(2006BAE01A01-11).

Synthesis and Insecticidal Activity of 2--1,3-dithiane Derivatives(Department of Applied Chemistry,China Agricultural University,Key Laboratory of PesticideChemistry and Application Technology,Beijing 100193,China)

  • 摘要: 为寻找新的环境友好型杀虫剂,用溴代呋喃甲醛和溴代噻吩甲醛分别与2-取代1,3-丙二硫醇缩合,合成了16个未见文献报道的2-溴代呋喃基或噻吩基-1,3-二噻烷衍生物。其化学结构均通过1H NMR和元素分析或质谱的确认。初步的生物活性测试结果表明,该类化合物对桃蚜Myzus persicae表现出一定的杀虫活性,其中化合物 M11 在600 μg/mL下对桃蚜的校正死亡率为90%。
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  • 收稿日期:  2008-05-01

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